REFERENCES

1. Bandini M, Eichholzer A. Catalytic functionalization of indoles in a new dimension. Angew Chem Int Ed Engl 2009;48:9608-44.

2. Kochanowska-Karamyan AJ, Hamann MT. Marine indole alkaloids: potential new drug leads for the control of depression and anxiety. Chem Rev 2010;110:4489-97.

3. Wan Y, Li Y, Yan C, Yan M, Tang Z. Indole: a privileged scaffold for the design of anti-cancer agents. Eur J Med Chem 2019;183:111691-708.

4. Maehr H, Smallheer J. Total syntheses of rivularins D1 and D3. J Am Chem Soc 1985;107:2943-5.

5. Zhang HH, Shi F. Organocatalytic atroposelective synthesis of indole derivatives bearing axial chirality: strategies and applications. Acc Chem Res 2022;55:2562-80.

6. Anilkumar GN, Lesburg CA, Selyutin O, et al. I. Novel HCV NS5B polymerase inhibitors: discovery of indole 2-carboxylic acids with C3-heterocycles. Bioorg Med Chem Lett 2011;21:5336-41.

7. Luz JG, Carson MW, Condon B, et al. Indole glucocorticoid receptor antagonists active in a model of dyslipidemia act via a unique association with an agonist binding site. J Med Chem 2015;58:6607-18.

8. Sharma K, Baral ER, Akhtar MS, Lee YR, Kim SH, Wee YJ. 3-Naphthylindoles as new promising candidate antioxidant, antibacterial, and antibiofilm agents. Res Chem Intermed 2017;43:2387-99.

9. Jiang F, Luo GZ, Zhu ZQ, Wang CS, Mei GJ, Shi F. Application of naphthylindole-derived phosphines as organocatalysts in[4 + 1] cyclizations of o-quinone methides with Morita-Baylis-Hillman carbonates. J Org Chem 2018;83:10060-9.

10. Li TZ, Liu SJ, Tan W, Shi F. Catalytic asymmetric construction of axially chiral indole-based frameworks: an emerging area. Chem Eur J 2020;26:15779-92.

11. Jiang F, Chen KW, Wu P, Zhang YC, Jiao Y, Shi F. A strategy for synthesizing axially chiral naphthyl-indoles: catalytic asymmetric addition reactions of racemic substrates. Angew Chem Int Ed Engl 2019;58:15104-10.

12. Sheng FT, Li ZM, Zhang YZ, et al. Atroposelective synthesis of 3,3’-bisindoles bearing axial and central chirality: using isatin-derived imines as electrophiles. Chin J Chem 2020;38:583-9.

13. Chen KW, Wang ZS, Wu P, et al. Catalytic asymmetric synthesis of 3,3’-bisindoles bearing single axial chirality. J Org Chem 2020;85:10152-66.

14. Qi LW, Mao JH, Zhang J, Tan B. Organocatalytic asymmetric arylation of indoles enabled by azo groups. Nat Chem 2018;10:58-64.

15. Zhu S, Chen YH, Wang YB, et al. Organocatalytic atroposelective construction of axially chiral arylquinones. Nat Commun 2019;10:4268-77.

16. Lu DL, Chen YH, Xiang SH, Yu P, Tan B, Li S. Atroposelective construction of arylindoles by chiral phosphoric acid-catalyzed cross-coupling of indoles and quinones. Org Lett 2019;21:6000-4.

17. Ding WY, Yu P, An QJ, et al. DFT-guided phosphoric-acid-catalyzed atroposelective arene functionalization of nitrosonaphthalene. Chem 2020;6:2046-59.

18. Chen YH, Li HH, Zhang X, Xiang SH, Li S, Tan B. Organocatalytic enantioselective synthesis of atropisomeric aryl-. p ;59:11374-8.

19. Zhang HH, Wang CS, Li C, Mei GJ, Li Y, Shi F. Design and enantioselective construction of axially chiral naphthyl-indole skeletons. Angew Chem Int Ed Engl 2017;56:116-21.

20. Bisag GD, Pecorari D, Mazzanti A, et al. Central-to-axial chirality conversion approach designed on organocatalytic enantioselective povarov cycloadditions: First access to configurationally stable indole-quinoline atropisomers. Chem Eur J 2019;25:15694-701.

21. He XL, Zhao HR, Song X, Jiang B, Du W, Chen YC. Asymmetric Barton-Zard reaction to access 3-pyrrole-containing axially chiral skeletons. ACS Catal 2019;9:4374-81.

22. Lu S, Ong JY, Yang H, et al. Diastereo- and atroposelective synthesis of bridged biaryls bearing an eight-membered lactone through an organocatalytic cascade. J Am Chem Soc 2019;141:17062-7.

23. Zhang X, Chen YH, Tan B. Organocatalytic enantioselective transformations involving quinone derivatives as reaction partners. Tetrahedron Lett 2018;59:473-86.

24. Chen YH, Qi LW, Fang F, Tan B. Organocatalytic atroposelective arylation of 2-naphthylamines as a practical approach to axially chiral biaryl amino alcohols. Angew Chem Int Ed Engl 2017;56:16308-12.

25. Cheng JK, Xiang SH, Tan B. Organocatalytic enantioselective synthesis of axially chiral molecules: development of strategies and skeletons. Acc Chem Res 2022;55:2920-37.

26. Kumarasamy E, Raghunathan R, Sibi MP, Sivaguru J. Nonbiaryl and heterobiaryl atropisomers: molecular templates with promise for atropselective chemical transformations. Chem Rev 2015;115:11239-300.

27. Cheng JK, Xiang SH, Li S, Ye L, Tan B. Recent advances in catalytic asymmetric construction of atropisomers. Chem Rev 2021;121:4805-902.

Chemical Synthesis
ISSN 2769-5247 (Online)

Portico

All published articles are preserved here permanently:

https://www.portico.org/publishers/oae/

Portico

All published articles are preserved here permanently:

https://www.portico.org/publishers/oae/